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API and intermediates
Products CAS No. Usage
 Diabetes
(R)-3-piperidinamine dihydrochloride 334618-23-4 Alogliptin intermediate
6-Chloro-3-methyluracil 4318-56-3 Alogliptin intermediate
6-Chlorouracil 4270-27-3 Alogliptin intermediate
2-[(6-Chloro-3,4-dihydro-3-Methyl-2,4-dioxo-1(2h)-pyriMidinyl)Methyl]benzonitrile 865758-96-9 Alogliptin intermediate
Alogliptin 850649-61-5 Alogliptin
Alogliptin Benzoate 850649-62-6 Alogliptin Benzoate
1,2-Diamino-2-methylpropane 811-93-8 Anagliptin intermediate
2-Methyl-1,2-propanediamine dihydrochloride 15444-85-6 Alogliptin intermediate
2-Methylpyrazolo[1,5-a]pyriMidine-6-carboxylic acid 739364-95-5 Anagliptin intermediate
(2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile 207557-35-5 Anagliptin intermediate
2,3,4,6-Tetrakis-O-trimethylsilyl-D-gluconolactone 32384-65-9 Canagliflozin intermediate
(5-bromo-2-Methylphenyl)(5-(4-fluorophenyl)thiophen-2-yl)Methanone 1132832-75-7 Canagliflozin intermidate
2-(5-bromo-2-methylbenzyl)-5-(4-fluorophenyl)thiophene 1030825-20-7 Canagliflozin intermediate
(5-(4-Fluorophenyl)thiophen-2-yl)(5-iodo-2-Methylphenyl)Methanone 1071929-08-2 Canagliflozin intermidate
2-(4-Fluorophenyl)-5-[(5-iodo-2-methylphenyl)methyl]thiophene 898566-17-1 Canagliflozin intermediate
Methyl 1-C-[3-[[5-(4-fluorophenyl)-2-thienyl]methyl]-4-methylphenyl]-D-glucopyranoside 1030825-21-8 Canagliflozin intermediate
(1S)-1,5-Anhydro-1-C-[3-[[5-(4-fluorophenyl)-2-thienyl]methyl]-4-methylphenyl]-D-glucitol tetraacetate 866607-35-4 Canagliflozin intermidate
Canagliflozin 842133-18-0 Canagliflozin
Canagliflozin Hemihydrate 928672-86-0 Canagliflozin Hemihydrate
2,3,4,6-Tetra-O-pivaloyl-alpha-D-glucopyranosyl bromide 81058-27-7 Dapagliflozin intermediate
5-bromo-2-chlorobenzoic acid 21739-92-4 Dapagliflozin intermediate
(5-bromo-2-chlorophenyl)(4-ethoxyphenyl)methanone 461432-22-4 Dapagliflozin intermediate
5-bromo-2-chloro-4’-ethoxydiphenylmethane 461432-23-5 Dapagliflozin intermediate
Methyl 1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-alpha-D-glucopyranoside 714269-57-5 Dapagliflozin intermediate
(1S)-1,5-Anhydro-1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-D-glucitol tetraacetate 461432-25-7 Dapagliflozin intermediate
2-Chloro-5-iodobenzoic acid 19094-56-5 Dapagliflozin intermediate
(5-Iodo-2-chlorophenyl)(4-ethoxyphenyl)methanone 1103738-26-6 Dapagliflozin intermediate
4-Iodo-1-chloro-2-(4-ethoxybenzyl)benzene 1103738-29-9 Dapagliflozin intermediate
Dapagliflozin 461432-26-8 Dapagliflozin
Dapagliflozin propanediol monohydrate 960404-48-2 Dapagliflozin propanediol monohydrate
4-[(5-Bromo-2-chlorophenyl)methyl]phenol 864070-18-8 Empagliflozin intermediate
(R)-tetrahydrofuran-3-yl 4-methylbenzenesulfonate 219823-47-9 Empagliflozin intermediate
(5-Bromo-2-chlorophenyl)[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methanone 915095-84-0 Ipragliflozin intermidate
(5-bromo-2-chlorophenyl)(4-fluorophenyl)methanone 915095-85-1 Empagliflozin intermediate
(3S)-3-[4-[(5-bromo-2-chlorophenyl)methyl]phenoxy]tetrahydrofuran 915095-89-5 Empagliflozin intermediate
(2S,3R,4S,5S,6R)-2-(3-(4-((S)-tetrahydrofuran-3-yloxy)benzyl)-4-chlorophenyl)-tetrahydro-6-(hydroxyMethyl)-2-Methoxy-2H-pyran-3,4,5-triol 1279691-36-9 Empagliflozin intermediate
(2-Chloro-5-iodophenyl)(4-fluorophenyl)methanone 915095-86-2 Empagliflozin intermediate
(2-Chloro-5-iodophenyl)[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methanone 915095-87-3 Empagliflozin intermediate
(3S)-3-[4-[(2-Chloro-5-iodophenyl)methyl]phenoxy]tetrahydro-furan 915095-94-2 Empagliflozin intermediate
(1S)-1,5-Anhydro-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydro-3-furanyl]oxy]phenyl]methyl]phenyl]-D-glucitol tetraacetate 915095-99-7 Empagliflozin intermidate
Empagliflozin 864070-44-0 Empagliflozin
Methyl 1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-5-C-(hydroxymethyl)-alpha-D-xylo-hexopyranoside 1528636-39-6 Ertugliflozin intermidate
Ertugliflozin 1210344-57-2 Ertugliflozin
Ertugliflozin L-pyroglutamic acid 1210344-83-4 Ertugliflozin L-pyroglutamic acid
2-Fluoro-5-Bromobenzaldehyde 93777-26-5 Ipragliflozin intermediate
2-(5-Bromo-2-fluorobenzyl)benzothiophene 1034305-17-3 Ipragliflozin intermediate
Ipragliflozin 761423-87-4 Ipragliflozin
Ipragliflozin L-proline 951382-34-6 Ipragliflozin L-proline
(R)-3-(Boc-Amino)piperidine 309956-78-3 Linagliptin intermediate
(S)-3-N-Boc-aminopiperidine 216854-23-8 Linagliptin intermediate
8-Bromo-3-methyl-xanthine 93703-24-3 Linagliptin intermediate
1-Bromo-2-butyne 3355-28-0 Linagliptin intermediate
8-bromo-7-(but-2-ynyl)-3-methyl-1H-purine-2,6(3H,7H)-dione 666816-98-4 Linagliptin intermediate
2-(chloromethyl)-4-methylquinazoline 109113-72-6 Linagliptin intermediate
8-Bromo-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydro-purine-2,6-dione 853029-57-9 Linagliptin intermidate
Boc Linagliptin 668273-75-4 Linagliptin intermidate
Linagliptin 668270-12-0 Linagliptin
Boc-3-Hydroxy-1-adamantyl-D-glycine 361442-00-4 Saxagliptin intermediate
(1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester 361440-67-7 Saxagliptin intermediate
(1S,3S,5S)-2-Azabicyclo[3.1.0]hexane-3-carboxamide mesylate 709031-45-8 Saxagliptin intermediate
Saxagliptin hydrate 945667-22-1 Saxagliptin hydrate
Saxagliptin hydrochloride 709031-78-7 NA
(5S)-4,5-O-(1-Methylethylidene)-1-C-4-morpholinyl-D-xylo-pentodialdo-5,2-furanose 1103738-19-7 Sotagliflozin intermidate
(5S)-1-C-[4-Chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-4,5-O-(1-methylethylidene)-D-xylo-pentodialdo-5,2-furanose 1103738-30-2 Sotagliflozin intermidate
Sotagliflozin 1018899-04-1 Sotagliflozin
Boc-(R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic acid 486460-00-8 Sitagliptin intermidate
3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride 762240-92-6 Sitagliptin intermidate
(2S)-4-Oxo-2-(3-thiazolidinylcarbonyl)-1-pyrrolidinecarboxylic acid tert-butyl ester 401564-36-1 Teneligliptin intermediate
Teneligliptin 760937-92-6 Teneligliptin
Teneligliptin Hydrobromide 906093-29-6 Teneligliptin Hydrobromide
Teneligliptin hydrobromide hydrate (2:5)X H2O 1572583-29-9 Teneligliptin hydrobromide hydrate (2:5)X H2O
2-CYANO-5-FLUOROBENZYL BROMIDE 421552-12-7 Trelagliptin (SYR472) intermediate
Trelagliptin 865759-25-7 Trelagliptin
Trelagliptin succinate 1029877-94-8 Trelagliptin (SYR472) succinate
2,3,4,6-Tetra-O-benzyl-D-glucono-1,5-lactone 13096-62-3 Tofogliflozin intermediate
2-Bromoterephthalic acid 586-35-6 Tofogliflozin intermediate
L-Prolinamide 7531-52-4 Vildagliptin intermediate
D-Prolinamide 62937-45-5 Vildagliptin intermediate
3-Amino-1-adamantanol 702-82-9 Vildagliptin intermediate
 Antiviral
3-Benzyloxy-4-oxo-4H-pyran-2-carboxylic acid 119736-16-2 Baloxavir intermediate
3-Benzyloxy-4-oxo-4H-pyran-2-carboxylic acid methyl ester 1332855-89-6 NA
(12aR)-3,4,12,12a-Tetrahydro-7-(phenylmethoxy)-1H-[1,4]oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione 1985607-70-2 Baloxavir intermediate
7,8-Difluoro-6,11-dihydrodibenzo[b,e]thiepin-11-ol 1985607-83-7 Baloxavir intermediate
3,4,12,12a-Tetrahydro-7-(phenylmethoxy)-1H-[1,4]oxazino[3,4-c]pyrido[2,1-f][1,2,4]triazine-6,8-dione 1370250-39-7 Balochavir intermediate
Chloromethyl methyl carbonate 40510-81-4 Baloxavir intermediate
7,8-Difluoro-dibenzo[b,e]thiepin-11(6H)-one 2136287-66-4 Baloxavir intermediate
3,4-DIFLUORO-2-METHYLBENZOIC ACID 157652-31-8 Baloxavir intermediate
Baloxavir 1985605-59-1 Baloxavir
Baloxavir marboxil 1985606-14-1 Baloxavir marboxil
3-Aminocyclopentanol hydrochloride 1184919-69-4 GS9883/Bictegravir intermidate
(1R,3S)-3-Aminocyclopentanol 1110772-05-8 Bictegravir intermediate
(1R,3S)-3-Aminocyclopentanol hydrochloride 1279032-31-3 Bictegravir intermediate
2,4,6-Trifluorobenzonitrile 96606-37-0 GS9883/Bictegravir intermediates
2,4,6-Trifluorobenzylamine 214759-21-4 Bictegravir intermediate
Bictegravir 1611493-60-7 Bictegravir
Bictegravir Sodium 1807988-02-8 Bictegravir Sodium
Phenyl hydrogen [(R)-1-(6-amino-9H-purin-9-yl)propan-2-yloxy]methylphosphonate 379270-35-6 Tenofovir alafenamide intermidate
Tenofovir alafenamide 379270-37-8 Tenofovir alafenamide
Tenofovir alafenamide Hemi-fumarate 1392275-56-7 Tenofovir alafenamide Hemi-fumarate
Tenofovir alafenamide fumarate 379270-38-9 Tenofovir alafenamide fumarate
 Antitumor
(3-Chloropyrazin-2-yl)MethanaMine hydrochloride 939412-86-9 Acalabrutinib intermidate
3-Chloropyrazin-2-methanamine dihydrochloride 867165-53-5 Acalabrutinib intermediate
(S)-Benzyl 2-(8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl)pyrrolidine-1-carboxylate 1420478-88-1 Acalabrutinib intermidate
N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide 1383385-64-5 Acalabrutinib intermidate
4-(PYRIDIN-2-YL)AMINOCARBONYLPHENYLBORONIC ACID 850568-25-1 Acalabrutinib intermidate
4-[8-Amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinylbenzamide 1420478-90-5 Acalabrutinib intermediate
Acalabrutinib /ACP-196 1420477-60-6 Acalabrutinib /ACP-196
(S)-(+)-3-Hydroxytetrahydrofuran 86087-23-2 Afatinib intermediate
(R)-(-)-3-Hydroxytetrahydrofuran 86087-24-3 Afatinib intermediate
Trans-4-Dimethylaminocrotonic acid hydrochloride 848133-35-7 Afatinib intermediate
7-Fluoro-6-nitro-4-hydroxyquinazoline 162012-69-3 Afatinib intermediate
Afatinib 439081-18-2/850140-72-6 Afatinib
Afatinib Dimaleate 850140-73-7 Afatinib Dimaleate
2-(Dimethylphosphinyl)benzenamine 1197953-47-1 Brigatinib intermidate
2,5-dichloro-N-(2-(diMethylphosphoryl)phenyl)pyriMidin-4-aMine 1197953-49-3 Brigatinib intermidate
1-[1-(3-methoxy-4-nitro-phenyl)-piperidin-4-yl]-4-methyl-piperazine 761440-65-7 Brigatinib intermidate
[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amine 761440-75-9 Brigatinib intermidate
Brigatinib 1197953-54-0 Brigatinib
(aR,3aS,4S,6S,7aR)-Hexahydro-3a,8,8-trimethyl-alpha-(2-methylpropyl)-4,6-methano-1,3,2-benzodioxaborole-2-methanamine 2,2,2-trifluoroacetate 179324-87-9 Bortezomib intermidate
N-(2-Pyrazinylcarbonyl)-L-phenylalanine 114457-94-2 Bortezomib intermidate
Bortezomib 179324-69-7 Bortezomib intermidate
3-Amino-4-cyano-5-(4-phenoxyphenyl)pyrazole 330792-70-6 Ibrutinib intermediate
5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine(N-2) 330786-24-8 Ibrutinib intermediate
(S)-1-Boc-3-hydroxypiperidine 143900-44-1 Ibrutinib intermediate
(R)-tert-Butyl 3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carboxylate (N-1) 1022150-11-3 Ibrutinib intermediate
3-(4-Phenoxy-phenyl)-1-piperidin-3-yl-1H-pyrazolo[3,4-d]pyrimidin-4-ylamine 1022150-12-4 Ibrutinib intermediate
Ibrutinib 936563-96-1 Ibrutinib
2-(2,5-Dichlorobenzamido)acetic acid 667403-46-5 Ixazomib (MLN9708)Intermediate
Ixazomib 1072833-77-2 Ixazomib
Ixazomib Citrate 1201902-80-8 Ixazomib (MLN9708) Citrate
Ixazomib citrate (USAN) 1239908-20-3 Ixazomib citrate (USAN)
4-Amino-3-chlorophenol 17609-80-2 Lenvatinib Intermediate
4-Amino-3-chlorophenol hydrochloride 52671-64-4 Lenvatinib intermediate
N-(2-Chloro-4-hydroxyphenyl)-N’-cyclopropyl-urea 796848-79-8 Lenvatinib intermediate
1,4-Dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester 205448-65-3 Lenvatinib intermidate
Methyl 4-chloro-7-methoxyquinoline-6-carboxylate 205448-66-4 Lenvatinib intermidate
4-Chloro-7-methoxyquinoline-6-carboxamide 417721-36-9 Lenvatinib intermidate
Lenvatinib 417716-92-8 Lenvatinib
Lenvatinib mesylate 857890-39-2 Lenvatinib mesylate
3-Hydroxyisobenzofuran-1(3h)-one 16859-59-9 Olaparib (AZD2281) intermediate
3-Oxo-1,3-dihydroisobenzofuran-1-ylphosphonic acid 61260-15-9 Olaparib (AZD2281) intermediate
2-FLUORO-5-FORMYLBENZONITRILE 218301-22-5 Olaparib (AZD2281) intermediate
2-Fluoro-5-[(3-oxo-1(3H)-isobenzofuranylidene)methyl]-benzonitrile 763114-25-6 Olaparib (AZD2281) intermediate
2-Fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)benzonitrile 1021298-68-9 Olaparib (AZD2281) intermediate
2-fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)Methyl)benzoic acid 763114-26-7 Olaparib Intermediate (AZD2281)
Tert-Butyl 4-(cyclopropanecarbonyl)piperazine-1-carboxylate 414910-15-9 Olaparib (AZD2281) intermediate
1-(Cyclopropylcarbonyl)piperazine 59878-57-8 Olaparib (AZD2281) intermediate
1-(cyclopropylcarbonyl)-, Monohydrochloride 1021298-67-8 Olaparib (AZD2281) intermediate
1-[5-[(3,4-Dihydro-4-oxo-1-phthalazinyl)methyl]-2-fluorobenzoyl]piperazine 763111-47-3 Olaparib intermediate
Olaparib 763113-22-0 Olaparib (AZD2281)
4-Fluoro-2-methoxy-5-nitroaniline 1075705-01-9 Osimertinib (AZD9291) intermediate
3-(2-Chloropyrimidin-4-yl)-1-meth ylindole 1032452-86-0 Osimertinib(AZD9291) intermediate
N,N,N’-TRIMETHYLETHYLENEDIAMINE 142-25-6 Osimertinib (AZD9291) intermediate
N1-[2-(Dimethylamino)ethyl]-5-methoxy-N1-methyl-N4-[4-(1-methyl-1H-indol-3-yl)-2-pyrimidinyl]-1,2,4-benzenetriamine 1421372-66-8 Osimertinib intermediates
Osimertinib 1421373-65-0 Osimertinib (AZD9291)
Osimertinib mesylate 1421373-66-1 Osimertinib mesylate
6-(Chloromethyl)uracil 18592-13-7 Tipiracil+Trifluridine/TAS-102 intermediate
2-AMINO-1-PYRROLINE HYDROCHLORIDE 7544-75-4 Tipiracil+Trifluridine/TAS-102 intermediate
5-(Trifluoromethyl)uracil 54-20-6 Tipiracil+Trifluridine/TAS-102 intermediate
Trifluridine 70-00-8 Trifluridine
 Cardiovascular
Ethyl chloro[(4-methoxyphenyl)hydrazono]acetate 27143-07-3 Apixaban intermidate
Ethyl (2Z)-chloro[(4-methoxyphenyl)hydrazono]ethanoate 473927-63-8 Apixaban intermidate
1-(4-Aminophenyl)-5,6-dihydro-3-(4-morpholinyl)-2(1H)-pyridinone 1267610-26-3 Apixaban intermidate
1-(4-IODO-PHENYL)-PIPERIDIN-2-ONE 385425-15-0 Apixaban intermidate
3-Chloro-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one 536760-29-9 Apixaban intermidate
3-(Morpholin-4-yl)-1-(4-nitrophenyl)-5,6-dihydropyridin-2(1H)-one 503615-03-0 Apixaban intermidate
3-Morpholin-4-yl-1-[4-(2-oxopiperidin-1-yl)phenyl]-5,6-dihydro-1H-pyridin-2-one 545445-44-1 Apixaban intermidate
4,5,6,7-Tetrahydro-1-(4-methoxyphenyl)-6-(4-nitrophenyl)-7-oxo-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid ethyl ester 536759-91-8 Apixaban intermidate
1-(4-Methoxyphenyl)-7-oxo-6-[4-(2-oxopiperidin-1-yl)phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid ethyl ester 503614-91-3 Apixaban intermidate
Apixaban 503612-47-3 Apixaban
2-Nitro-5-methoxybenzoic acid 1882-69-5 Betrixaban intermidate
2-Amino-5-methoxybenzoic acid 6705-03-9 Betrixaban intermidate
Betrixaban 330942-05-7 Betrixaban
Betrixaban Maleate 936539-80-9 Betrixaban Maleate
2-THIOADENOSINE 43157-50-2 Cangrelor intermediate
CLODRONIC ACID 10596-23-3 Cangrelor Intermediate
CLODRONIC ACID N-BUTYLAMINE SALT 163706-61-4 Cangrelor intermediate
2-CHLOROETHYL METHYL SULFIDE 542-81-4 Cangrelor intermediate
(2R,3R,4S,5R)-2-(6-aMino-2-(3,3,3-trifluoropropylthio)-9H-purin-9-yl)-5-(hydroxyMethyl)tetrahydrofuran-3,4-diol 163706-51-2 Cangrelor intermediate
(2R,3S,4R,5R)-2-(hydroxyMethyl)-5-(6-((2-(Methylthio)ethyl)aMino)-2-((3,3,3-trifluoropropyl)thio)-9H-purin-9-yl)tetrahydrofuran-3,4-diol 163706-58-9 Cangrelor intermediate
Cangrelor base 163706-06-7 Cangrelor base
Cangrelor tetrasodium 163706-36-3 Cangrelor tetrasodium
4,5,6,7-tetrahydro-5-Methyl-Thiazolo[5,4-c]pyridin 720720-96-7 Edoxaban intermediate
[(5-Chloro-2-pyridinyl)amino]oxoacetic acid 552850-73-4 Edoxaban intermediate
N-(5-chloro-pyridin-2-yl)-oxalamic acid ethyl ester 349125-08-2  Edoxaban intermediate
2-[(5-Chloropyridin-2-yl)amino]-2-oxoacetic acid ethyl ester monohydrochloride 1243308-37-3 Edoxaban intermediate
(S)-(-)-3-Cyclohexenecarboxylic acid 5708-19-0 Edoxaban intermediate
(1S,3R,4R)-3-(Boc-aMino)-4-hydroxy-cyclohexanecarboxylic acid ethyl ester 365997-33-7 Edoxaban intermediate
(1S,3S,6R)-N,N-dimethyl-7-oxabicyclo[4.1.0]heptane-3-carboxamide 929693-35-6 Edoxaban intermidate
Tert-Butyl [(1R,2S,5S)-2-amino-5-[(dimethylamino)carbonyl]cyclohexyl]carbamate 365998-36-3 Edoxaban Intermediate
Tert-Butyl(1R,2S,5S)-2-azido-5-[(dimethylamino)carbonyl]cyclohexylcarbamate oxalic acid 1210348-34-7 Edoxaban intermediate
Tert-Butyl(1R,2S,5S)-2-azido-5-[(dimethylamino)carbonyl]cyclohexylcarbamate oxalic acid monohydrate 1353893-22-7 Edoxaban intermediate
Edoxaban 480449-70-5 Edoxaban
Edoxaban tosylate 480449-71-6/912273-65-5 Edoxaban tosylate
Edoxaban tosylate monohydrate 1229194-11-9 Edoxaban tosylate monohydrate
5-Isoquinolinesulfonic acid 27655-40-9 Fasudil HCl intermidate
ISOQUINOLINE-5-SULFONYL CHLORIDE 84468-15-5 Fasudil HCl intermidate
Isoquinoline-5-sulphonyl chloride hydrochloride 105627-79-0 Fasudil HCl intermidate
Homopiperazine 505-66-8 Fasudil HCL 中间体
FASUDIL 103745-39-7 Fasudil
Fasudil HCl 105628-07-7 Fasudil HCl
(R)-tert-butyl-(1-([1,1’-biphenyl]-4-yl)-3-hydroxypropan-2-yl)carbamate 1426129-50-1 Sacubitril/AHU-377 /LCZ696 intermediate
(R,E)-5-([1,1’-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2-Methylpent-2-enoic acid 1012341-48-8 Sacubitril/ AHU-377/LCZ696 intermediate
(2R,4S)-5-(Biphenyl-4-yl)-4-[(tert-butoxycarbonyl)amino]-2-methylpentanoic acid 1012341-50-2 Sacubitril/ AHU-377 /LCZ696 intermediate
(2R,4S)-4-Amino-5-(biphenyl-4-yl)-2-methylpentanoic acid ethyl ester hydrochloride 149690-12-0 Sacubitril/AHU-377 /LCZ696 Intermediate
Sacubitril 149709-62-6 Sacubitril/ AHU -377/ LCZ696
AHU-377 hemicalcium salt (2:1) 1369773-39-6 AHU-377 hemicalcium salt (2:1)
LCZ696 936623-90-4 LCZ696
5-Chloro-2-thiophenecarboxylic acid 24065-33-6 Rivaroxaban intermediate
5-Chlorothiophene-2-carbonyl chloride 42518-98-9 Rivaroxaban intermidate
4-(4-aminophenyl)morpholin-3-one 438056-69-0 Rivaroxaban intermediate
(S)-(+)-N-(2,3-Epoxypropyl)phthalimide 161596-47-0 Rivaroxaban intermediate
2-[(2R)-2-HYDROXY-3-[[4-(3-OXO-4-MORPHOLINYL)PHENYL]AMINO]PROPYL]-1H-ISOINDOLE-1,3(2H)-DIONE 446292-07-5 Rivaroxaban intermediate
2-({(5S)-2-oxo-3-[4-(3-oxomorpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl} 446292-08-6 Rivaroxaban intermediate
4-[4-[(5S)-5-(Aminomethyl)-2-oxo-3-oxazolidinyl]phenyl]-3-morpholinone hydrochloride 898543-06-1 Rivaroxaban intermediate
Rivaroxaban 366789-02-8 Rivaroxaban
5-Chloro-2,3-diphenylpyrazine 41270-66-0 Selexipag intermediate
4-[(1-Methylethyl)amino]-1-butanol 42042-71-7 Selexipag intermediate
4-[(5,6-Diphenylpyrazinyl)(1-methylethyl)amino]-1-butanol 475086-75-0 Selexipag intermediate
Selexipag 475086-01-2 Selexipag
 Other categories
4-Chloropyrrolo[2,3-d]pyrimidine 3680-69-1 Baricitinib intermediate
4-Chloro-7-[[2-(trimethylsilyl)ethoxy]methyl]-7H-pyrrolo[2,3-d]pyrimidine 941685-26-3 Baricitinib intermediate
1-(1-Ethoxyethyl)-1H-pyrazole-4-boronic acid pinacol ester 1029716-44-6 Baricitinib intermediate
4-(1H-Pyrazol-4-yl)-7-[[2-(trimethylsilyl)ethoxy]methyl]-7H-pyrrolo[2,3-d]pyrimidine 941685-27-4 Baricitinib intermediate
Tert-Butyl 3-oxoazetidine-1-carboxylate 398489-26-4 Baricitinib intermediate
3-(Cyanomethylene)-1-azetidinecarboxylic acid tert-butyl ester 1153949-11-1 Baricitinib intermediate
2-[1-(Ethylsulfonyl)-3-azetidinylidene]acetonitrile 1187595-85-2 Baricitinib intermediate
(4-(1-(3-(cyanomethyl)-1-(ethylsulfonyl)azetidin-3-yl)-1H-pyrazol-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl pivalate 1187595-90-9 Baricitinib intermediate
Baricitinib 1187594-09-7 Baricitinib
Baricitinib phosphate salt 1187595-84-1 Baricitinib phosphate salt
3-benzyl-6-bromo-2-chloroquinoline 654655-68-2 Bedaquiline intermediate
3-Benzyl-6-bromo-2-methoxyquinoline 654655-69-3 Bedaquiline intermediate
3-(Dimethylamino)-1-(naphthalen-1-yl)propan-1-one 10320-49-7 Bedaquiline intermediate
3-Dimethylamino-1-(naphthalen-1-yl)propan-1-one hydrochloride 5409-58-5 Bedaquiline intermediate
(R)-(-)-1,1’-Binaphthyl-2,2’-diyl hydrogenphosphate 39648-67-4 Bedaquiline intermediate
Bedaquiline 843663-66-1 Bedaquiline
Bedaquiline fumarate 845533-86-0 Bedaquiline fumarate
2-Bromo-5-hydroxybenzaldehyde 2973-80-0 Crisaborole (AN-2728 intermediate
4-[4-Bromo-3-(1,3-dioxolan-2-yl)phenoxy]benzonitrile 1217366-74-9 Crisaborole (AN-2728)intermediate
4-(4-Bromo-3-formylphenoxy)benzonitrile 906673-54-9 Crisaborole (AN-2728)intermediate
4-[4-Bromo-3-(hydroxymethyl)phenoxy]benzonitrile 906673-45-8 Crisaborole (AN-2728)intermediate
4-(3-Formylphenoxy)benzonitrile 90178-72-6 Crisaborole (AN-2728)intermediate
Crisaborole 906673-24-3 Crisaborole (AN-2728)
(5S)-5-Phenyl-2-morpholinone hydrochloride 491833-36-4 Eliglustat intermediate
1,4-Benzodioxane-6-carboxaldehyde 29668-44-8 Eliglustat intermediate
(1R,3S,5S,8aS)-1,3-Bis(2,3-dihydro-1,4-benzodioxin-6-yl)tetrahydro-5-phenyl-3H,8H-oxazolo[4,3-c][1,4]oxazin-8-one 491833-25-1 Eliglustat intermediate
1-[(2S,3R)-3-(2,3-Dihydro-1,4-benzodioxin-6-yl)-3-hydroxy-2-[[(1S)-2-hydroxy-1-phenylethyl]amino]-1-oxopropyl]pyrrolidine 491833-26-2 Eliglustat intermediate
(1R,2R)-2-Amino-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-(pyrrolidin-1-yl)propan-1-ol 491833-28-4 Eliglustat intermediate
2,5-Dioxopyrrolidin-1-yl octanoate 14464-30-3 Eliglustat intermediate
Eliglustat 491833-29-5 Eliglustat
Eliglustat tartrate 928659-70-5 Eliglustat tartrate
(S)-1-(5-PHENYL-1H-IMIDAZOL-2-YL)ETHANAMINE 864825-23-0 Eluxadoline intermediate
Methyl 5-formyl-2-methoxybenzoate 78515-16-9 Eluxadoline intermediate
4-(Aminocarbonyl)-N-[(1,1-dimethylethoxy)carbonyl]-2,6-dimethyl-L-phenylalanine 623950-02-7 Eluxadoline intermediate
Eluxadoline 864821-90-9 Eluxadoline
Eluxadoline Dihydrochloride 864825-13-8 Eluxadoline Dihydrochloride
Thiomorpholine-1,1-dioxide 39093-93-1 Filgotinib intermidate
Thiomorpholine-1,1-dioxide hydrochloride 59801-62-6 Filgotinib intermediate
5-Chloro[1,2,4]triazolo[1,5-a]pyridin-2-amine 175965-64-7 Filgotinib intermidate
5-Bromo-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine 1010120-55-4 Filgotinib intermidate
N-(5-Bromo[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide 1142943-96-1 Filgotinib intermidate
Filgotinib 1206161-97-8 Filgotinib
Filgotinib maleate 1802998-75-9 Filgotinib maleate
1 ,3-dimethyl adamantane 702-79-4 Memantine intermediate
1-Bromo-3,5-dimethyladamantane 941-37-7 Memantine intermediate
Memantine HCI 41100-52-1 Memantine HCI
Imidazo[1,2-a]pyridin-3-ylacetic acid 17745-04-9 Minodronic acid intermidate
Ethyl (E)-4,4-dimethoxy-2-butenoate 114736-25-3 Minodronic acid intermediate
Minodronic acid 180064-38-4 Minodronic acid
4-Nitrophenethylamine hydrochloride 29968-78-3 Mirabegron intermediate
(alphaR)-alpha-[[[2-(4-Nitrophenyl)ethyl]amino]methyl]benzenemethanol hydrochloride 521284-21-9 Mirabegron intermediate
(alphaR)-alpha-[[[2-(4-Aminophenyl)ethyl]amino]methyl]benzenemethanol hydrochloride 521284-22-0 Mirabegron intermediate
2-Aminothiazol-4-acetic acid 29676-71-9 Mirabegron intermediate
Mirabegron 223673-61-8 Mirabegron
N-Ethyl-N-methyl carbamoyl chloride 42252-34-6 Rivastigmine intermediate
3-(1-(dimethylamino)ethyl)phenol 105601-04-5 Rivastigmine intermediate
(S)-3-(1-(dimethylamino)ethyl)phenol 139306-10-8 Rivastigmine intermediate
Rivastigmine 123441-03-2 Rivastigmine
Rivastigmine tartrate 129101-54-8 Rivastigmine tartrate
4-Amino-3-hydroxybenzoic acid 2374-03-0 Tafamidis intermediate
3,5-Dichlorobenzoyl chloride 2905-62-6 Tafamidis intermediate
3,5-Dichlorobenzoic acid 51-36-5 Tafamidis intermediate
Tafamidis 594839-88-0 Tafamidis
Tafamidis meglumine 951395-08-7 Tafamidis meglumine
2,4-Dichloro-1H-pyrrolo[2,3-d]pyrimidine 90213-66-4 Tofacitinib intermediate
N,4-Dimethyl-1-(phenylmethyl)-3-piperidinamine hydrochloride (1:2) 1228879-37-5 Tofacitinib intermediate
(3R,4R)-1-Benzyl-N,4-dimethylpiperidin-3-amine 477600-70-7 Tofacitinib intermediate
(3R,4R)-N,4-Dimethyl-1-(phenylmethyl)-3-piperidinamine hydrochloride 1062580-52-2 Tofacitinib intermediate
(2R,3R)-2,3-Bis[(4-methylbenzoyl)oxy]butanedioic acid compd. with (3R,4R)-N,4-dimethyl-1-(phenylmethyl)-3-piperidinamine 477600-71-8 Tofacitinib intermidate
N-Methyl-N-[(3R,4R)-4-methyl-1-(phenylmethyl)-3-piperidinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine 477600-73-0 Tofacitinib intermediate
cis-1-Benzyl-N-methyl-4-methylpiperidin-3-amine dihydrochloride 477600-68-3
N-methyl-N-((3R,4R)-4-methylpiperidin-3-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (N-1 BASE) 477600-74-1 Tofacitinib intermediate
N-Methyl-N-((3R,4R)-4-Methylpiperidin-3-yl)-7H-pyrrolo[2,3-d]pyriMidin-4-amine dihydrochloride (N-1 HCl) 1260590-51-9 Tofacitinib intermediate
Tofacitinib BASE 477600-75-2 Tofacitinib BASE
Tofacitinib Citratet 540737-29-9 Tofacitinib Citratet
2,6-Dichlorobenzyl bromide 20443-98-5 Vilanterol intermidate
2-bromo-1-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-Ethanone 102293-80-1 Vilanterol intermidate
tert-butyl 2-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-2-oxoethylcarbamate 452339-71-8 Vilanterol intermidate
tert-butyl (2R)-2-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-2-hydroxyethylcarbamate 452339-72-9 Vilanterol intermidate
5-(2,2-diMethyl-4H-benzo[d][1,3]dioxin-6-yl)oxazolidin-2-one 452340-96-4 Vilanterol intermidate
(5R)-5-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)-1,3-oxazolidin-2-one 452339-73-0 Vilanterol intermidate
2-[(2,6-Dichlorophenyl)methoxy]-ethanol 85309-91-7 Vilanterol intermidate
Benzene, 2-[[2-[(6-broMohexyl)oxy]ethoxy]Methyl]-1,3-dichloro 503070-57-3 Vilanterol intermidate
(5R)-3-[6-[2-[(2,6-dichlorophenyl)Methoxy]ethoxy]hexyl]-5-(2,2-diMethyl-4H-1, 3-benzodioxin-6-yl)-2-Oxazolidinone 503068-36-8 Vilanterol intermidate
(1R)-2-[[6-[2-[(2,6-Dichlorobenzyl)oxy]ethoxy]hexyl]amino]-1-(2,2-dimethyl-4H-1,3-benzodioxin-6-yl)ethanol 503068-37-9 Vilanterol intermidate
Triphenylacetic acid 595-91-5 Vilanterol intermidate
Vilanterol 503068-34-6 Vilanterol
Vilanterol Trifenate 503070-58-4 Vilanterol Trifenate
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